Year Winner Institution Title Journal Full author list
2016 Ayo Egunlusi University of the Western Cape Tricycloundecane Derivatives as Potential N-Methyl­D-aspartate (NMDA) Receptor and Voltage-Gated Calcium Channel Modulators ChemMedChem Sarel Malan, Jacques Joubert
2015 Frank Zindo University of the Western Cape Polycyclic propargylamine and acetylene derivatives as multifunctional neuroprotective agents European Journal of Medicinal Chemistry Quinton Barber, Jacques Joubert, Jacobus Bergh, Jacobus Petzer and Sarel Malan
2014 Dr Ilze Vermaak Tshwane University of Technology Hyperspectral imaging in the quality control of herbal medicines – The case of neurotoxic Japanese star anise Journal of Pharmaceutical and Biomedical Analysis Alvaro Viljoen and Susanne Lindström
2013 Prof Sarel Malan University of the Western Cape and North West University S-Nitrosylation and Attentuation of Excessive Calcium Flux Pentacycloundecane Derivatives Medicinal Chemistry, 2012, 8, 361-371 Hendrik Lemmer, Jacques Joubert, Sandra van Dyk and Francois van der Westhuizen
2012 Dr Jacques Joubert School of Pharmacy, University of the Western Cape Synthesis, evaluation and application of polycyclic fluorescent analogues as N­methyl-D-aspartate receptor and voltage gated calcium channel ligands European Journal of Medicinal Chemistry 46 (2011) 5010-5020
2011 Belinda Strydom School of Pharmacy, North West University – Potchefstroom campus Inhibition of monoamine oxidase by 8-benzylcaffeine analogues Bioorganic and Medicinal Chemistry 18: 1018–1028 SF Malan, N Castagnoli, JJ Bergh and JP Petzer
2010 Sarel F Malan School of Pharmacy, University of the Western Cape Synthesis and in vitro evaluation of pteridine analogues as monoamine oxidase B and nitric oxide synthase inhibitors Bio-organic and Medicinal Chemistry
2009 Jacobus J Bergh School of Pharmacy, North West University – Potchefstroom campus Structure-activity relationships in the inhibition of monoamine oxidase B by 1­methyl-3 phenylpyrroles Bio-organic and Medicinal Chemistry Ogunrombi MO, Malan SF, Terreblanche G, Castagnoli Jr N, Bergh JJ, Petzer JP
2008 Jacobus P Petzer School of Pharmacy, North West University – Potchefstroom campus Inhibition of monoamine oxidase B by selected benzimidazole and caffeine analogues Bioorganic and Medicinal Chemistry 15 (2007) 3692-3702 Deidré vd Berg, Kevin Zoellner, Modupe Ogunrombi, Sarel Malan, Gisella Terre’Blanche, Neal Castagnoli and Jacobus Bergh
2007 Sarel F Malan School of Pharmacy, North West University – Potchefstroom campus Inhibition of monoamine oxidase B by analogues of the adenosine A2A receptor antagonist (E)-8-(3­chlorostyryl) caffeine (CSC) Bioorganic and Medicinal Chemistry 14 (2006) 3512-3521 Nevil Vlok, Neal Castagnoli Jr, Cobus Bergh and Jacobus Petzer
2006 Alvaro Viljoen School of Pharmacy, Tshwane University of Technology The composition, geographical variation and antimicrobial activity of Lippia javanica (Verbenaceae) leaf essential oils Journal of Ethnopharmacology 2005: 96: 271-277 S Subramoney, SF van Vuuren, KHC Baser and B Demirci
2005 Sarel F Malan School of Pharmacy, North West University – Potchefstroom campus Fluorescent ligands for the histamine H2 receptor: synthesis and preliminary characterization Bioorganic and Medicinal Chemistry (2004) 12: 6495-6503 Sarel F Malan, Andre van Marle, Wiro M Menge, Valentine Zuliana, Marcel Hoffman, Henk Timmerman and Rob Leurs
2004 Jaco Zah School of Pharmacy, North West University – Potchefstroom campus Physicochemical Prediction of a Brain-Blood Distribution Profile in Polycyclic Amines Bioorganic & Medicinal Chemistry (2003) 11: 3569-3578 Jaco Zah, Gisella Terre’Blanche, Elardus Erasmus and Sarel F Malan
2003 Sarel F Malan School of Pharmacy, Potchefstroom University for CHE Antimalarial compounds from Parinari capensis Bioorganic and Medicinal Chemistry Letters (2002). 12: 2167-2169 Arina C Uys, Sarel F Malan, Sandra van Dyk and Robyn L van Zyl
2002 Theunis C Goosen School of Pharmacy, Potchefstroom University for CHE Effects of Benzyl Isothiocyanate on Rat and human Cytochromes P450 : Identification of metabolites formed by P450 2B1 Journal of Pharmacology and Experimental Therapeutics (2001) 296(1): 198-206 Theunis C Goosen, Danielle E Mills and Paul F Hollenberg
2001 Sarel F Malan School of Pharmacy, Potchefstroom University for CHE Structure-Activity Relationships of Polycyclic Aromatic Amines with Calcium Channel Blocking Activity Arch. Pharm. Pharm. Med. Chem.(2000) 333:10-16 Sarel F Malan, Jurgens van der Walt and Cornelius J van der Schyf
2000 Mino R Caira University of Cape Town Resolution of Albuterol Acetonide Tetrahedron: Asymmetry (1999) 10: 2175-2189 Mino R Caira, R Hunter, Luigi R Nassimbeni and Anne T Stevens
1999 Sarel F Malan School of Pharmacy, Potchefstroom University for CHE
1998 Kobus Bergh School of Pharmacy, Potchefstroom University for CHE
1997 Kobus Bergh School of Pharmacy, Potchefstroom University for CHE
1996 Douglas W Oliver School of Pharmacy, Potchefstroom University for CHE
1995 Douglas W Oliver School of Pharmacy, Potchefstroom University for CHE
1994 Mino R Caira University of Cape Town